Structural basis for partial agonism in 5-HT3A receptors
Kevin Felt, Madeleine Stauffer, Leslie Salas-Estrada, Peter R. Guzzo, Dejian Xie, Jinkun Huang, Marta Filizola, Sudha Chakrapani
Topics & Concepts
Partial agonistNauseaIrritable bowel syndromeVomitingReceptorSerotoninPharmacology5-HT receptorChemistryAntagonistMedicineInternal medicinePharmacogenetics and Drug MetabolismReceptor Mechanisms and SignalingPhenothiazines and Benzothiazines Synthesis and Activities