Litcius/Paper detail

Combining radial and continuous flow synthesis to optimize and scale-up the production of medicines

Mara Guidi, Sooyeon Moon, Lucia Anghileri, Dario Cambié, Peter H. Seeberger, Kerry Gilmore

2021Reaction Chemistry & Engineering26 citationsDOIOpen Access PDF

Abstract

Rapid, standardized process optimization and development on a radial synthesizer can be directly converted to a dedicated continuous flow process for scale-up, shown for three APIs <italic>via</italic> single- and multistep syntheses and continuous crystallization.

Topics & Concepts

Continuous flowScale (ratio)Process engineeringContinuous productionProcess (computing)Computer scienceFlow (mathematics)MathematicsEngineeringBiochemical engineeringChemical engineeringPhysicsProgramming languageGeometryQuantum mechanicsInnovative Microfluidic and Catalytic Techniques InnovationAnalytical Chemistry and ChromatographyCrystallization and Solubility Studies
Combining radial and continuous flow synthesis to optimize and scale-up the production of medicines | Litcius