Design and synthesis of 1,4-disubstituted 1,2,3-triazoles: Biological evaluation, in silico molecular docking and ADME screening
İrfan Şahin, Mustafa Çeşme, Fatma Betül Özgeriş, Özge Güngör, Ferhan Tümer
Topics & Concepts
ChemistryDPPHPropargylAscorbic acidABTSAcarboseAntioxidantTroloxHeLaADMEDocking (animal)IC50NaringinStereochemistryOrganic chemistryEnzymeNuclear chemistryChromatographyBiochemistryIn vitroCatalysisFood scienceNursingMedicineClick Chemistry and ApplicationsComputational Drug Discovery MethodsSynthesis and biological activity