Discovery of a AHR pelargonidin agonist that counter-regulates Ace2 expression and attenuates ACE2-SARS-CoV-2 interaction
Michele Biagioli, Silvia Marchianò, Rosalinda Roselli, Cristina Di Giorgio, Rachele Bellini, Martina Bordoni, Anna Gidari, Samuele Sabbatini, Daniela Francisci, Bianca Fiorillo, Bruno Catalanotti, Eleonora Distrutti, Adriana Carino, Angela Zampella, Gabriele Costantino, Stefano Fiorucci
Topics & Concepts
Downregulation and upregulationAryl hydrocarbon receptorInflammationReceptorAngiotensin-converting enzyme 2PharmacologyBiologyImmunologyChemistryInternal medicineBiochemistryMedicineTranscription factorDiseaseCoronavirus disease 2019 (COVID-19)Infectious disease (medical specialty)GeneCOVID-19 Clinical Research StudiesSARS-CoV-2 and COVID-19 ResearchLong-Term Effects of COVID-19