Discovery of the first Mycobacterium tuberculosis MabA (FabG1) inhibitors through a fragment-based screening
Léo Faïon, Kamel Djaout, Rosangela Frita, Catalin Pintiala, François‐Xavier Cantrelle, Martin Moune, Alexandre Vandeputte, Kévin Bourbiaux, Catherine Piveteau, Adrien Herlédan, Alexandre Biela, Florence Leroux, Laurent Kremer, Mickaël Blaise, Abdalkarim Tanina, René Wintjens, Xavier Hanoulle, Benoît Déprez, Nicolas Willand, Alain R. Baulard, Marion Flipo
Topics & Concepts
INHAMycobacterium tuberculosisAnthranilic acidEnzymeBiochemistryChemistryDocking (animal)TuberculosisBiologyMedicineNursingPathologyTuberculosis Research and EpidemiologyMicrobial Natural Products and BiosynthesisBiochemical and Molecular Research