Dose-dependent bioavailability and tissue distribution of the ATR inhibitor AZD6738 (ceralasertib) in mice
Brian F. Kiesel, Jianxia Guo, Robert A. Parise, Raman Venkataramanan, David A. Clump, Christopher J. Bakkenist, Jan H. Beumer
Topics & Concepts
BioavailabilityPharmacokineticsPharmacologyCamptothecinDistribution (mathematics)DNA damageDrugMetabolismImmune systemMetaboliteBiologyImmunologyDNAEndocrinologyBiochemistryMathematical analysisMathematicsDNA Repair MechanismsCarcinogens and Genotoxicity AssessmentPARP inhibition in cancer therapy