Design, synthesis and biological evaluation of novel phenylfuran-bisamide derivatives as P-glycoprotein inhibitors against multidrug resistance in MCF-7/ADR cell
Zhikun Yang, Xue Yang, Yasheng Li, Yue Cai, Yanlei Yu, Wenya Zhuang, Xuanrong Sun, Qingyong Li, Xiaoze Bao, Xinyi Ye, Jin‐Miao Tian, Bin Wei, Jianwei Chen, Qihao Wu, Huawei Zhang, Xiaozhou Mou, Hong Wang
Topics & Concepts
ChemistryP-glycoproteinMultiple drug resistanceEffluxCytotoxicityPharmacologyIC50Rhodamine 123Lead compoundDocking (animal)StereochemistryIn vitroBiochemistryMedicineAntibioticsNursingDrug Transport and Resistance MechanismsCancer therapeutics and mechanismsHIV/AIDS drug development and treatment