Litcius/Paper detail

Design, synthesis and biological evaluation of novel phenylfuran-bisamide derivatives as P-glycoprotein inhibitors against multidrug resistance in MCF-7/ADR cell

Zhikun Yang, Xue Yang, Yasheng Li, Yue Cai, Yanlei Yu, Wenya Zhuang, Xuanrong Sun, Qingyong Li, Xiaoze Bao, Xinyi Ye, Jin‐Miao Tian, Bin Wei, Jianwei Chen, Qihao Wu, Huawei Zhang, Xiaozhou Mou, Hong Wang

2023European Journal of Medicinal Chemistry26 citationsDOI

Topics & Concepts

ChemistryP-glycoproteinMultiple drug resistanceEffluxCytotoxicityPharmacologyIC50Rhodamine 123Lead compoundDocking (animal)StereochemistryIn vitroBiochemistryMedicineAntibioticsNursingDrug Transport and Resistance MechanismsCancer therapeutics and mechanismsHIV/AIDS drug development and treatment