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Design, synthesis and molecular docking of novel substituted azepines as inhibitors of PI3K/Akt/TSC2/mTOR signaling pathway in colorectal carcinoma

Ahmed A. Noser, Aboubakr H. Abdelmonsef, Maha M. Salem

2022Bioorganic Chemistry36 citationsDOI

Topics & Concepts

PI3K/AKT/mTOR pathwayProtein kinase BChemistryCancer researchKinaseDocking (animal)In silicoSignal transductionBiochemistryBiologyGeneMedicineNursingPI3K/AKT/mTOR signaling in cancerSynthesis and Biological ActivityQuinazolinone synthesis and applications
Design, synthesis and molecular docking of novel substituted azepines as inhibitors of PI3K/Akt/TSC2/mTOR signaling pathway in colorectal carcinoma | Litcius