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Drugging the undruggable RAS: Mission Possible?

Adrienne D. Cox, Stephen W. Fesik, Alec C. Kimmelman, Ji Luo, Channing J. Der

2014Nature Reviews Drug Discovery2,012 citationsDOIOpen Access PDF

Topics & Concepts

EffectorComputational biologyBiologyBioinformaticsComputer scienceCell biologyProtein Kinase Regulation and GTPase SignalingPI3K/AKT/mTOR signaling in cancerProtein Degradation and Inhibitors
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