Synthesis of indazoles from 2-formylphenylboronic acids
Vitalii V. Solomin, Alberts Seins, Aigars Jirgensons
Abstract
A method for the synthesis of indazoles was developed which involves a copper(<sc>ii</sc>) acetate catalysed reaction of 2-formylboronic acids with diazadicaboxylates followed by acid or base induced ring closure.
Topics & Concepts
ChemistryCombinatorial chemistryChemical Synthesis and AnalysisClick Chemistry and ApplicationsSynthesis of Indole Derivatives