Safety, pharmacokinetics, and antiretroviral activity of islatravir (ISL, MK-8591), a novel nucleoside reverse transcriptase translocation inhibitor, following single-dose administration to treatment-naive adults infected with HIV-1: an open-label, phase 1b, consecutive-panel trial
Dirk Schürmann, Deanne Jackson Rudd, Saijuan Zhang, Inge De Lepeleire, Martine Robberechts, Evan Friedman, Christian Keicher, Andreas Hüser, Jörg Hofmann, Jay A. Grobler, S. Aubrey Stoch, Marian Iwamoto, Randolph P. Matthews
Topics & Concepts
MedicinePharmacokineticsReverse-transcriptase inhibitorTolerabilityDosingNucleoside Reverse Transcriptase InhibitorAdverse effectPharmacologyInternal medicineLamivudineExpanded accessViral loadImmunologyHuman immunodeficiency virus (HIV)VirusAntiretroviral therapyHepatitis B virusHIV/AIDS drug development and treatmentHIV Research and TreatmentHIV-related health complications and treatments