Saikosaponins and the deglycosylated metabolites exert liver meridian guiding effect through PXR/CYP3A4 inhibition
Qiwei Liu, Yunwen Xue, Jingjing Liu, Siqi Ren, Jie Xu, Jinni Yang, Yuanyue Xing, Zunjian Zhang, Rui Song
Topics & Concepts
CYP3A4MicrosomePharmacologyChemistryIC50BiochemistryMetabolismIn vitroBiologyCytochrome P450Pharmacogenetics and Drug MetabolismNatural product bioactivities and synthesisFlavonoids in Medical Research