Chalcone Mannich base derivatives: synthesis, antimalarial activities against <i>Plasmodium knowlesi</i>, and molecular docking analysis
Jufrizal Syahri, Rahmiwati Hilma, Amatul Hamizah Ali, Norzila Ismail, Ng Yee Ling, Nurlaili Nurlaili, Beta Achromi Nurohmah, Hani Kartini Agustar, Lau Yee Ling, Jalifah Latip
Abstract
Research on the antimalarial effect of aminoalkyl chalcone derivatives against Plasmodium falciparum and Plasmodium knowlesi has bolstered efforts in drug discovery to combat cases of drug resistance.
Topics & Concepts
ChalconePlasmodium falciparumChemistryPlasmodium knowlesiStereochemistryMannich baseAntimalarial AgentCombinatorial chemistryOrganic chemistryBiologyMalariaImmunologyPlasmodium vivaxMalaria Research and ControlSynthesis and biological activityResearch on Leishmaniasis Studies