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WaterMap and Molecular Dynamic Simulation-Guided Discovery of Potential PAK1 Inhibitors Using Repurposing Approaches

Jayashree Biswal, Prajisha Jayaprakash, Suresh K. Rayala, Ganesh Venkatraman, Raghu Rangaswamy, Jeyaraman Jeyakanthan

2021ACS Omega21 citationsDOIOpen Access PDF

Abstract

analysis.

Topics & Concepts

DrugBankChemistryDocking (animal)Molecular dynamicsDrug repositioningDrugDrug discoveryPharmacologySmall moleculeBiochemistryComputational chemistryBiologyMedicineNursingComputational Drug Discovery MethodsProtein Kinase Regulation and GTPase SignalingEnzyme Structure and Function
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