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Discovery of ML210-Based glutathione peroxidase 4 (GPX4) degrader inducing ferroptosis of human cancer cells

Han Wang, Chao Wang, Bingru Li, Cangxin Zheng, Guoquan Liu, Zhenming Liu, Liangren Zhang, Ping Xu, Ping Xu

2023European Journal of Medicinal Chemistry55 citationsDOIOpen Access PDF

Topics & Concepts

GPX4ChemistryLysosomeCancer cellAutophagyHT1080Lipid peroxidationGlutathione peroxidaseCancerGlutathioneCell biologyCancer researchBiochemistryCellOxidative stressEnzymeApoptosisBiologyGeneticsFerroptosis and cancer prognosisHistone Deacetylase Inhibitors ResearchPeptidase Inhibition and Analysis
Discovery of ML210-Based glutathione peroxidase 4 (GPX4) degrader inducing ferroptosis of human cancer cells | Litcius