Litcius/Paper detail

Recent advances in EZH2-based dual inhibitors in the treatment of cancers

Xiaojuan Yang, Xu Lu, Yang Li

2023European Journal of Medicinal Chemistry27 citationsDOIOpen Access PDF

Topics & Concepts

EZH2ChemistryMethyltransferasePRC2HistoneCancer researchHistone methyltransferaseHistone H3Small moleculeIn vivoMethylationBiologyBiochemistryGeneticsDNAEpigenetics and DNA MethylationHistone Deacetylase Inhibitors ResearchProtein Degradation and Inhibitors