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Novel guanidine derivatives targeting leukemia as selective Src/Abl dual inhibitors: Design, synthesis and anti-proliferative activity

Amr H. Moustafa, Asmaa M. AboulMagd, Ali M. Ali, A. Khodairy, Adel A. Marzouk, Ayman Nafady, Mohamed T. M. Nemr

2024Bioorganic Chemistry27 citationsDOI

Topics & Concepts

ChemistryIC50Proto-oncogene tyrosine-protein kinase SrcABLKinaseTyrosine kinaseMAPK/ERK pathwayStereochemistryBiochemistrySignal transductionIn vitroChronic Myeloid Leukemia TreatmentsQuinazolinone synthesis and applicationsResearch on Leishmaniasis Studies
Novel guanidine derivatives targeting leukemia as selective Src/Abl dual inhibitors: Design, synthesis and anti-proliferative activity | Litcius