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Collateral lethality between HDAC1 and HDAC2 exploits cancer-specific NuRD complex vulnerabilities

Yuxiang Zhang, David Remillard, Ugoma Onubogu, Barbara Karakyriakou, Joshua N. Asiaban, Anissa R. Ramos, Kirsten Bowland, Timothy R. Bishop, Paige Barta, Stephanie Nance, Adam D. Durbin, Christopher J. Ott, Michalina Janiszewska, Benjamin F. Cravatt, Michael A. Erb

2023Nature Structural & Molecular Biology34 citationsDOIOpen Access PDF

Topics & Concepts

BiologyChromatinHistone deacetylase 2Histone deacetylaseHDAC1EnhancerHistoneGeneticsChromatin remodelingCancer researchCell biologyTranscription factorComputational biologyGeneHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsUbiquitin and proteasome pathways
Collateral lethality between HDAC1 and HDAC2 exploits cancer-specific NuRD complex vulnerabilities | Litcius