Exploiting polypharmacology to dissect host kinases and kinase inhibitors that modulate endothelial barrier integrity
Selasi Dankwa, Mary-Margaret Dols, Ling Wei, Elizabeth K. K. Glennon, Heather S. Kain, Alexis Kaushansky, Joseph D. Smith
Topics & Concepts
KinaseDrug discoveryBiologyDrug repositioningCell biologyPharmacologyDrugBioinformaticsComputational Drug Discovery MethodsProtein Kinase Regulation and GTPase SignalingReceptor Mechanisms and Signaling