Computationally guided discovery of novel non-steroidal AR-GR dual antagonists demonstrating potency against antiandrogen resistance
Xin Chai, Xueping Hu, Xinyue Wang, Huating Wang, Jinping Pang, Wenfang Zhou, Jianing Liao, Luhu Shan, Xiaohong Xu, Lei Xu, Hongguang Xia, Tingjun Hou, Dan Li
Topics & Concepts
Androgen receptorAntiandrogenAntagonistProstate cancerAndrogen Receptor AntagonistsPharmacologyIC50PotencyChemistryMedicineReceptorInternal medicineIn vitroCancerBiochemistryProstate Cancer Treatment and ResearchEstrogen and related hormone effectsReceptor Mechanisms and Signaling