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A potent new-scaffold androgen receptor antagonist discovered on the basis of a MIEC-SVM model

Xinyue Wang, Xin Chai, Luhu Shan, Xiaohong Xu, Lei Xu, Tingjun Hou, Huiyong Sun, Dan Li

2024Acta Pharmacologica Sinica10 citationsDOIOpen Access PDF

Topics & Concepts

Androgen receptorAntagonistScaffoldAndrogenComputational biologyReceptorChemistryPharmacologyBiologyComputer scienceInternal medicineMedicineEndocrinologyHormoneProstate cancerDatabaseCancerProstate Cancer Treatment and ResearchHormonal and reproductive studiesReceptor Mechanisms and Signaling
A potent new-scaffold androgen receptor antagonist discovered on the basis of a MIEC-SVM model | Litcius