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Aroyl Fluorides as Bifunctional Reagents for Dearomatizing Fluoroaroylation of Benzofurans

Xiaoye Yu, Qingyuan Meng, Constantin G. Daniliuc, Armido Studer

2022Journal of the American Chemical Society163 citationsDOIOpen Access PDF

Abstract

-acylated indoles to afford 3-aroyl-2-fluoro-dihydroindoles.

Topics & Concepts

ChemistryBifunctionalReagentOrganic chemistryCombinatorial chemistryCatalysisFluorine in Organic ChemistryRadical Photochemical ReactionsSulfur-Based Synthesis Techniques
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