Litcius/Paper detail

New scaffolds for type II JAK2 inhibitors overcome the acquired G993A resistance mutation

Matthew L. Arwood, Yao Liu, Shannon Harkins, David M. Weinstock, Lei Yang, Kristen E. Stevenson, Olivia D. Plana, Jingyun Dong, Haley Cirka, Kristen L. Jones, Anniina Virtanen, Dikshat Gopal Gupta, Amanda Ceas, Brian Lawney, Akinori Yoda, Catharine Leahy, Mingfeng Hao, Zhixiang He, Hwan Geun Choi, Yaning Wang, Olli Silvennoinen, Stevan R. Hubbard, Tinghu Zhang, Nathanael S. Gray, Loretta S. Li

2023Cell chemical biology12 citationsDOIOpen Access PDF

Topics & Concepts

MutationCancer researchSmall moleculeKinasePolycythemia veraIn vivoJanus kinase 2ChemistryMedicineBiologyBiochemistryGeneGeneticsImmunologyMyeloproliferative Neoplasms: Diagnosis and TreatmentCytokine Signaling Pathways and InteractionsChronic Myeloid Leukemia Treatments