Synthesis of novel pyrazino[1,2-a]indol-1(2H)-one derivatives as potent cholinesterase inhibitors and their in vitro and in silico evaluations
Burak Kuzu, Yeliz Demir
Topics & Concepts
ButyrylcholinesteraseTacrineCholinesteraseIn silicoAcetylcholinesteraseChemistryDocking (animal)PharmacologyAchéDonepezilDrug discoveryEnzymeBiochemistryStereochemistryComputational biologyBiologyMedicineDementiaNursingPathologyDiseaseGeneCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsSynthesis and biological activity