Litcius/Paper detail

Discovery of new 1 <i>H</i> -pyrazolo[3,4- <i>d</i> ]pyrimidine derivatives as anticancer agents targeting EGFR <sup>WT</sup> and EGFR <sup>T790M</sup>

Ahmed A. Abdel Gaber, Mohamed Sobhy, Abdallah Turky, Hanan Gaber Abdulwahab, Ahmed A. Al‐Karmalawy, Mostafa A. Elhendawy, Mohamed. M. Radwan, Eslam B. Elkaeed, Ibrahim M. Ibrahim, Heba S. A. Elzahabi, Ibrahim H. Eissa

2022Journal of Enzyme Inhibition and Medicinal Chemistry44 citationsDOIOpen Access PDF

Abstract

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Topics & Concepts

PyrimidineChemistryT790MStereochemistryCombinatorial chemistryEpidermal growth factor receptorBiochemistryGefitinibReceptorLung Cancer Treatments and MutationsSynthesis and biological activityPI3K/AKT/mTOR signaling in cancer