Medicinal chemistry strategies to discover P-glycoprotein inhibitors: An update
Jinyun Dong, Zuodong Qin, Weidong Zhang, Gang Cheng, Assaraf G. Yehuda, Charles R. Ashby, Zhe‐Sheng Chen, Xiangdong Cheng, Jiang‐Jiang Qin
Topics & Concepts
P-glycoproteinEffluxMultiple drug resistanceATP-binding cassette transporterPharmacologyClinical trialToxicityCancer cellCancerDrugChemotherapyMedicineChemistryTransporterCancer researchInternal medicineAntibioticsBiochemistryGeneDrug Transport and Resistance MechanismsPharmacological Effects and Toxicity StudiesHIV/AIDS drug development and treatment