Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications
Nicholas Favalli, Gabriele Bassi, Christian Pellegrino, Jacopo Millul, Roberto De Luca, Samuele Cazzamalli, Su Yang, Anika Trenner, Nour L. Mozaffari, Renier Myburgh, Mustafa Moroglu, Stuart J. Conway, Alessandro A. Sartori, Markus G. Manz, Richard A. Lerner, Peter K. Vogt, Jörg Scheuermann, Dario Neri
Topics & Concepts
ChemistryDNAComputational biologyLigand (biochemistry)Drug discoveryRegioselectivityCombinatorial chemistryChemical librarySmall moleculeBiochemistryReceptorCatalysisBiologyMonoclonal and Polyclonal Antibodies ResearchClick Chemistry and ApplicationsProtein Degradation and Inhibitors