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The Problems of Applying Classical Pharmacology Analysis to Modern In Vitro Drug Discovery Assays: Slow Binding Kinetics and High Target Concentration

Sam R.J. Hoare

2021SLAS DISCOVERY30 citationsDOIOpen Access PDF

Topics & Concepts

Drug discoveryPotencyDrugComputational biologyChemistryLigand efficiencyLead compoundPharmacologyIn vitroLigand (biochemistry)BioassayDrug developmentCombinatorial chemistryBiophysicsBiochemistryBiologyReceptorGeneticsComputational Drug Discovery MethodsMonoclonal and Polyclonal Antibodies ResearchReceptor Mechanisms and Signaling
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