Discovery of new anticancer thiourea-azetidine hybrids: design, synthesis, in vitro antiproliferative, SAR, in silico molecular docking against VEGFR-2, ADMET, toxicity, and DFT studies
Deepa R. Parmar, Jigar Y. Soni, Ramakrishna Guduru, Rahul H. Rayani, Rakesh V. Kusurkar, Anand Vala, Sahista N. Talukdar, Ibrahim H. Eissa, Ahmed M. Metwaly, Ahmed Khalil, Vishwanath Zunjar, Satyanarayana Battula
Topics & Concepts
ChemistryAzetidineA431 cellsStereochemistryDocking (animal)Cell cultureDU145In silicoIn vitroCisplatinBiochemistryCancer cellCellCell cycleCancerBiologyLNCaPGeneticsMolecular medicineMedicineChemotherapyNursingGeneSynthesis of β-Lactam CompoundsSynthesis and Catalytic ReactionsClick Chemistry and Applications