Litcius/Paper detail

Are the current commercially available oximes capable of reactivating acetylcholinesterase inhibited by the nerve agents of the A-series?

Marcelo C. dos Santos, Fernanda D. Botelho, Arlan da Silva Gonçalves, Daniel A. S. Kitagawa, Caio Borges, Taynara Carvalho-Silva, Leandro B. Bernardo, Cíntia N. Ferreira, Rafael B. Rodrigues, Denise Cristian Ferreira Neto, Eugenie Nepovimová, Kamil Kuča, Steven R. LaPlante, Antônio Luís dos Santos Lima, Tanos C. C. França, Samir F. A. Cavalcante

2022Archives of Toxicology28 citationsDOI

Topics & Concepts

AcetylcholinesteraseNerve agentOximeIn silicoAchéDocking (animal)ChemistryPharmacologyCombinatorial chemistryStereochemistryBiochemistryEnzymeBiologyMedicineVeterinary medicineGeneCholinesterase and Neurodegenerative DiseasesPesticide Exposure and ToxicityComputational Drug Discovery Methods