A deep learning-based theoretical protocol to identify potentially isoform-selective PI3Kα inhibitors
Muhammad Shafiq, Zaid Anis Sherwani, Mamona Mushtaq, Mohammad Nur‐e‐Alam, Aftab Ahmad, Zaheer Ul‐Haq
Topics & Concepts
ADMEIn silicoComputational biologyPI3K/AKT/mTOR pathwayDocking (animal)Small moleculeDrug discoveryBinding affinitiesChemistryDrugPharmacologyBiologyBiochemistrySignal transductionReceptorMedicineGeneNursingPI3K/AKT/mTOR signaling in cancerClick Chemistry and ApplicationsBiochemical and Molecular Research