Litcius/Paper detail

σ-Bond initiated generation of aryl radicals from aryl diazonium salts

Elene Tatunashvili, Bun Chan, Philippe E. Nashar, Christopher S. P. McErlean

2020Organic & Biomolecular Chemistry31 citationsDOI

Abstract

σ-Bond nucleophiles and molecular oxygen transform aryl diazonium salts into aryl radicals. Experimental and computational studies show that Hantzsch esters transfer hydride to aryl diazonium species, and that oxygen initiates radical fragmentation of the diazene intermediate to produce aryl radicals. The operational simplicity of this addition-fragmentation process for the generation of aryl radicals, by a polar-radical crossover mechanism, has been illustrated in a variety of bond-forming reactions.

Topics & Concepts

ChemistryRadicalArylAryl radicalDiazonium CompoundsOxygenPhotochemistryOrganic chemistryPolymer chemistryAlkylRadical Photochemical ReactionsSulfur-Based Synthesis TechniquesCatalytic C–H Functionalization Methods