Design, synthesis and biological evaluation of a novel spiro oxazolidinedione as potent p300/CBP HAT inhibitor for the treatment of ovarian cancer
Hong Ding, Yuan Pei, Yuan‐Qing Li, Wen Xu, Lianghe Mei, Zeng Hou, Yiman Guang, Liyuan Cao, Peizhuo Li, Haijing Cao, Jinlei Bian, Kaixian Chen, Cheng Luo, Bing Zhou, Ting Zhang, Zhiyu Li, Yaxi Yang
Topics & Concepts
AcetylationChemistryEpigeneticsHistoneOvarian cancerCarcinogenesisCancer researchChromatinCancerBiochemistryBiologyGeneticsDNAGeneHistone Deacetylase Inhibitors ResearchUbiquitin and proteasome pathwaysProtein Degradation and Inhibitors