BRET- and fluorescence anisotropy-based assays for real-time monitoring of ligand binding to M2 muscarinic acetylcholine receptors
Lukas Grätz, Tõnis Laasfeld, Anni Allikalt, Corinna G. Gruber, Andrea Pegoli, Maris‐Johanna Tahk, Mari-Liis Tsernant, Max Keller, Ago Rinken
Topics & Concepts
Muscarinic acetylcholine receptorFluorescenceLigand (biochemistry)RadioligandChemistryLigand binding assayBinding siteBiophysicsFluorescence anisotropyRadioligand AssayReceptorReceptor–ligand kineticsBinding affinitiesG protein-coupled receptorBiochemistryBiologyMembraneQuantum mechanicsPhysicsReceptor Mechanisms and SignalingPharmacological Effects and AssaysNicotinic Acetylcholine Receptors Study