Discovery of harmiprims, harmine-primaquine hybrids, as potent and selective anticancer and antimalarial compounds
Kristina Pavić, Goran Poje, Laís Pessanha de Carvalho, Tana Tandarić, Marina Marinović, Diana Fontinha, Jana Held, Miguel Prudêncio, Ivo Piantanida, Robert Vianello, I. Kneževic, Ivana Perković, Zrinka Rajić
Topics & Concepts
ChemistryHarmineCancer cellPrimaquineAntimalarial AgentPlasmodium falciparumCell cycleBiochemistryCell cycle checkpointPharmacologyStereochemistryCellCancerChloroquineMalariaBiologyGeneticsImmunologySynthesis and bioactivity of alkaloidsCancer therapeutics and mechanismsSynthesis and Biological Evaluation