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Gardenin B, A Natural Inhibitor for USP7: <i>In vitro</i> Evaluation and <i>In silico</i> Identification

Siyu Zhang, Yujie Sun, Zhongyue Bai, Yifan Wang, Guangjian Zhao, Fengli Yao, Yacong Yang, Yu Hu, Xionghao Li, Fang Liu, Peng Wang, Peng Wang, Ximing Xu

2023Letters in Drug Design & Discovery12 citationsDOI

Topics & Concepts

Deubiquitinating enzymeIn silicoChemistryNatural productIn vitroEnzymeUbiquitinIC50Active siteDocking (animal)CytotoxicityComputational biologyBiochemistryBiologyGeneMedicineNursingUbiquitin and proteasome pathways