Synthesis, biological evaluation, Structure − Activity relationship studies of quinoline-imidazole derivatives as potent antimalarial agents
Deblina Roy, Mohammad Anas, Ashan Manhas, Satyen Saha, Niti Kumar, Gautam Panda
Topics & Concepts
ChemistryQuinolinePlasmodium falciparumEnantiomerImidazoleAntimalarial AgentStereochemistrySelectivityIC50CytotoxicityCombinatorial chemistryBiological activityIn vitroBiochemistryMalariaOrganic chemistryCatalysisBiologyImmunologyMalaria Research and ControlPhenothiazines and Benzothiazines Synthesis and ActivitiesComputational Drug Discovery Methods