Synthesis and inhibitory activity of euparin derivatives as potential dual inhibitors against α-glucosidase and protein tyrosine phosphatase 1B (PTP1B)
Jinqiang Wang, Dandan Feng, Yimin Xiang, Ji Guo, Nianyu Huang, Na Yu, Huishu Yang, Cheng‐Xiong Liu, Kun Zou
Topics & Concepts
ChalconeNatural productIC50Protein tyrosine phosphataseBiochemistryChemistryEnzymeDocking (animal)AcarbosePhosphataseLead compoundPharmacologyStereochemistryBiologyIn vitroMedicineNursingNatural product bioactivities and synthesisNatural Antidiabetic Agents StudiesCarbohydrate Chemistry and Synthesis