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Dual inhibitors of HDAC and other epigenetic regulators: A novel strategy for cancer treatment

Ekta Shirbhate, Vaibhav Singh, Varsha Jahoriya, Aditya Mishra, Ravichandran Veerasamy, Amit K. Tiwari, Harish Rajak

2023European Journal of Medicinal Chemistry34 citationsDOIOpen Access PDF

Topics & Concepts

EpigeneticsHistoneEpigenetic therapyHistone deacetylaseCancer epigeneticsDrug discoveryComputational biologyChemistryDNA methylationBiologyPharmacologyBioinformaticsGeneGeneticsGene expressionHistone methyltransferaseHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsEpigenetics and DNA Methylation
Dual inhibitors of HDAC and other epigenetic regulators: A novel strategy for cancer treatment | Litcius