Design, synthesis, and biological evaluation of new 2-(4-(methylsulfonyl)phenyl)-N-phenylimidazo[1,2-a]pyridin-3-amine as selective COX-2 inhibitors
Mahsa Azami Movahed, Fatemeh Abbası, Mahsa Rajabi, Niusha Abedi, Nima Naderi, Bahram Daraei, Afshin Zarghi
Topics & Concepts
ChemistryPharmacophoreStereochemistryAmine gas treatingActive siteSelectivityEnzymeHydrogen bondArachidonate 5-lipoxygenaseArachidonic acidMoleculeOrganic chemistryCatalysisSynthesis and biological activityInflammatory mediators and NSAID effectsSynthesis and Reactions of Organic Compounds