Litcius/Paper detail

Biosynthesis of the Prenylated Salicylaldehyde Flavoglaucin Requires Temporary Reduction to Salicyl Alcohol for Decoration before Reoxidation to the Final Product

Jonas Nies, Huomiao Ran, Viola Wohlgemuth, Wen‐Bing Yin, Shu‐Ming Li

2020Organic Letters35 citationsDOI

Abstract

The biosynthetic pathway of the prenylated salicylaldehyde flavoglaucin and congeners in Aspergillus ruber was elucidated by genome mining, heterologous expression, precursor feeding, and biochemical characterization. The polyketide skeleton was released as alkylated salicyl alcohols, which is a prerequisite for consecutive hydroxylation and prenylation, before reoxidation to the final aldehyde products. Our results provide an excellent example for a highly programmed machinery in natural product biosynthesis.

Topics & Concepts

PrenylationChemistrySalicylaldehydeBiosynthesisNatural productPolyketideHydroxylationAldehydeAlcoholCombinatorial chemistryStereochemistryOrganic chemistryCatalysisEnzymeSchiff baseMicrobial Natural Products and BiosynthesisPlant biochemistry and biosynthesisNatural product bioactivities and synthesis