Design and synthesis of novel coumarin derivatives as potential acetylcholinesterase inhibitors for Alzheimer's disease
Kamilia M. Amin, Doaa E. Abdel Rahman, Heba Abdelrasheed Allam, Haidy H. El-Zoheiry
Topics & Concepts
ChemistryAcetylcholinesteraseAcetamideCoumarinIC50Docking (animal)StereochemistryActive siteEnzymeDonepezilIn vivoIn silicoIn vitroBiochemistryOrganic chemistryGeneDiseaseDementiaBiologyMedicinePathologyNursingBiotechnologyCholinesterase and Neurodegenerative DiseasesSynthesis and biological activityComputational Drug Discovery Methods