Development of CVN424: A Selective and Novel GPR6 Inverse Agonist Effective in Models of Parkinson Disease
Nicola Brice, Hans H. Schiffer, Holger Monenschein, Victoria Mulligan, Keith J. Page, Justin Powell, Xiao Xu, Toni Cheung, J. Russell Burley, Huikai Sun, Louise Dickson, Sean T. Murphy, Nidhi Kaushal, Steve Sheardown, Jason Lawrence, Yun Chen, Darian M. Bartkowski, Anne Kanta, Joseph Russo, Natalie Hosea, Lee A. Dawson, Stephen Hitchcock, Mark Carlton
Topics & Concepts
StriatumAgonistDopaminergicParkinson's diseasePharmacologyMedium spiny neuronSubstantia nigraInverse agonistReceptorNeuroscienceMedicineDopamineChemistryInternal medicineBiologyDiseaseReceptor Mechanisms and SignalingNeuroscience and Neuropharmacology ResearchNeurotransmitter Receptor Influence on Behavior