Litcius/Paper detail

Development of CVN424: A Selective and Novel GPR6 Inverse Agonist Effective in Models of Parkinson Disease

Nicola Brice, Hans H. Schiffer, Holger Monenschein, Victoria Mulligan, Keith J. Page, Justin Powell, Xiao Xu, Toni Cheung, J. Russell Burley, Huikai Sun, Louise Dickson, Sean T. Murphy, Nidhi Kaushal, Steve Sheardown, Jason Lawrence, Yun Chen, Darian M. Bartkowski, Anne Kanta, Joseph Russo, Natalie Hosea, Lee A. Dawson, Stephen Hitchcock, Mark Carlton

2021Journal of Pharmacology and Experimental Therapeutics43 citationsDOI

Topics & Concepts

StriatumAgonistDopaminergicParkinson's diseasePharmacologyMedium spiny neuronSubstantia nigraInverse agonistReceptorNeuroscienceMedicineDopamineChemistryInternal medicineBiologyDiseaseReceptor Mechanisms and SignalingNeuroscience and Neuropharmacology ResearchNeurotransmitter Receptor Influence on Behavior