Design, syntheses and evaluations of novel indole derivatives as orally selective estrogen receptor degraders (SERD)
Jiaqiang Dong, Tie-lin Wang, Jianyu Lu, Charles Z. Ding, Lihong Hu, Guoping Hu, Huijun He, Xu Zeng, Xiaoting Li, Deheng Sun, Yingjie Zhu, Liang Shen, Qingyang Gu, Chi-Chung Chan, Yuanfeng Xia, Jian Li, Shuhui Chen
Topics & Concepts
FulvestrantEstrogen receptorChemistryPharmacologyBreast cancerIndole testIn vivoEstrogen receptor alphaBioavailabilityCancerSelective estrogen receptor modulatorCancer researchInternal medicineStereochemistryMedicineBiologyBiotechnologyEstrogen and related hormone effectsHER2/EGFR in Cancer ResearchClick Chemistry and Applications