Design, synthesis and biological evaluation of novel HDAC inhibitors with improved pharmacokinetic profile in breast cancer
Dahong Yao, Chenyang Li, Jin Jiang, Jian Huang, Jinhui Wang, Zhendan He, Jin Zhang
Topics & Concepts
ChemistryAcetylationPharmacokineticsHistone deacetylasePharmacologyApoptosisEpigeneticsAutophagyBiochemistryHistoneBiologyGeneHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsCholinesterase and Neurodegenerative Diseases