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Highly selective inhibitors of protein kinases CLK and HIPK with the furo[3,2-b]pyridine core

Václav Němec, Lukáš Maier, Benedict‐Tilman Berger, A. Chaikuad, Stanislav Drápela, Karel Souček, Stefan Knapp, Kamil Paruch

2021European Journal of Medicinal Chemistry32 citationsDOIOpen Access PDF

Topics & Concepts

PharmacophoreChemistryPyridineChemical biologyKinaseStereochemistryChemical synthesisDrug discoveryCombinatorial chemistryBiochemistryIn vitroMedicinal chemistryBiochemical and Molecular ResearchSynthesis and Reactivity of HeterocyclesChronic Lymphocytic Leukemia Research
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