Discovery of natural alkaloids as potent and selective inhibitors against human carboxylesterase 2
Yi‐Shu Zhao, Xing‐Kai Qian, Xiao‐Qing Guan, Pei‐Fang Song, Yun‐Qing Song, Rong-Jing He, Mengru Sun, Xiu-Yang Wang, Li‐Wei Zou, Guang‐Bo Ge
Topics & Concepts
ChemistryCarboxylesteraseButyrylcholinesteraseReserpinePharmacologySerineBiochemistryBenzimidazoleNon-competitive inhibitionSerine hydrolaseEnzymeStereochemistryAcetylcholinesteraseMedicineAchéOrganic chemistryCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsSynthesis and bioactivity of alkaloids